Exam questionKROK 1Dentistry · 2018
A patient with dislocated jaw was given a short-acting muscle relaxant by a doctor. Name this drug:
Answer options
- Cytitonum (Cytisine)
- Dithylinum (Suxamethonium chloride)
- Procaine
- Papaverine hydrochloride
- Pyridostigmine hydrobromide
Correct answer
Dithylinum (Suxamethonium chloride)
Explanation
Muscle relaxants1. Non-depolarizing muscle relaxant:• Tubocurarine (Curariform)Mechanism: blockage of N-cholinergic receptors of the synaptic membraneAntidote: Proserin (Neostigmine)2. Depolarizing muscle relaxant:Curarelike Dithylinum (Suxamethonium)Mechanism:Over-depolarized N-cholinergic receptors =Muscle is overstimulatedThen, muscle desensitize (muscle desensitization).That’s why it cause muscle contraction at the beginning.Antidote:Acetylcholinesterase by blood transfusion
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